Detailed comparison of Tirzepatide and Retatrutide — mechanisms, dosing, side effects, costs, and best use cases.
| Factor | Tirzepatide | Retatrutide |
|---|---|---|
| Category | GLP-1 / Weight Loss | GLP-1 / Weight Loss |
| Common Dose | 2,500–15,000 mcg | 4,000–12,000 mcg |
| Frequency | Once weekly | Once weekly |
| Half-Life | ~5 days | ~6 days |
| Best For | FDA-approved, proven safety profile, currently widely available | Maximum weight loss in clinical trials, Phase 3 trials ongoing |
GLP-1 / Weight Loss
Tirzepatide (Mounjaro/Zepbound) is the first dual GIP/GLP-1 receptor agonist, producing superior weight loss vs semaglutide — averaging 20–22% body weight reduction in the SURMOUNT trials. By activating both GIP and GLP-1 receptors, it enhances insulin sensitivity, reduces appetite via dual hypothal...
Dose: 2,500–15,000 mcg
Frequency: Once weekly
⚡ Tirzepatide CalculatorGLP-1 / Weight Loss
Retatrutide is a next-generation triple agonist targeting GIP, GLP-1, and glucagon receptors simultaneously — the most powerful weight loss compound in clinical development. Phase 2 trials by Eli Lilly demonstrated up to 24% body weight reduction, exceeding both semaglutide (~15%) and tirzepatide (~...
Dose: 4,000–12,000 mcg
Frequency: Once weekly
⚡ Retatrutide CalculatorRetatrutide's triple mechanism (GIP+GLP-1+Glucagon) shows ~24% weight loss in Phase 2 vs tirzepatide's ~22%. However, retatrutide is not yet FDA-approved.
Tirzepatide (Mounjaro/Zepbound) is the first dual GIP/GLP-1 receptor agonist, producing superior weight loss vs semaglutide — averaging 20–22% body weight reduction in the SURMOUNT trials. By activating both GIP and GLP-1 receptors, it enhances insulin sensitivity, reduces appetite via dual hypothalamic pathways, slows gastric emptying, and improves beta-cell function. FDA-approved for type 2 diabetes (Mounjaro) and weight management (Zepbound). Starting dose: 2.5 mg weekly, titrated every 4 weeks to 15 mg maximum. Track your tirzepatide titration schedule with the DoseIQ app.
📖 Read Full Tirzepatide Dosing Guide →Retatrutide is a next-generation triple agonist targeting GIP, GLP-1, and glucagon receptors simultaneously — the most powerful weight loss compound in clinical development. Phase 2 trials by Eli Lilly demonstrated up to 24% body weight reduction, exceeding both semaglutide (~15%) and tirzepatide (~22%). Adding glucagon receptor activation further increases energy expenditure and fatty acid oxidation. Currently in Phase 3 trials; FDA approval expected 2026–2027. Compounded research versions available.
📖 Read Full Retatrutide Dosing Guide →The #1 peptide tracking app for iPhone. Calculate doses, log injections, set reminders, and track your progress.
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